Small molecule NNMT inhibitor (non-peptide), 5-amino-1-methylquinolinium Technical specifications
Before injection (preparation phase) 30 minutes before: Remove tirzepatide from the refrigerator to reach room temperature 15 minutes before: Gather supplies: alcohol swabs, cold pack, hydrocortisone cream, clean needle 1 hour before: Take oral antihistamine (cetirizine 10mg) if you have a history of reactions Choose injection site: Check your log for the last site used
Combination therapy should only be done under a doctors supervision
Update, June 29, 2026: After this piece first published, the FDA posted its briefing documents for the July meeting, and its own reviewers proposed not to add BPC-157, in either of its chemical forms, to the compounding list
However, this medication isn't recommended for individuals with a family or personal history of medullary thyroid carcinoma or Multiple Endocrine Neoplasia syndrome type 2
PMC 7899277